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BR103
CAS No. 1434873-26-3
BR103( BR 103 )
Catalog No. M11848 CAS No. 1434873-26-3
BR103 is a potent, metabolically stable and highly selective small molecule agonist of complement C3a receptor (C3aR) with EC50 of 22 ± 8 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 873 | In Stock |
|
| 50MG | 1782 | In Stock |
|
| 100MG | 2250 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBR103
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NoteResearch use only, not for human use.
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Brief DescriptionBR103 is a potent, metabolically stable and highly selective small molecule agonist of complement C3a receptor (C3aR) with EC50 of 22 ± 8 nM.
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DescriptionBR103 is a potent, metabolically stable and highly selective small molecule agonist of complement C3a receptor (C3aR) with EC50 of 22 ± 8 nM; displays high selectivity for C3aR over C5aR; induces paw oedema and mast cell activation in vivo in rats.
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In Vitro——
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In Vivo——
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SynonymsBR 103
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PathwayImmunology/Inflammation
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TargetComplement System
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RecptorComplement System
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Research Area——
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Indication——
Chemical Information
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CAS Number1434873-26-3
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Formula Weight448.527
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Molecular FormulaC24H28N6O3
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Purity>98% (HPLC)
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Solubility——
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SMILESN=C(N)NCCC[C@@H](C(O)=O)NC(C1=C(C)NC(C(C2=CC=CC=C2)C3=CC=CC=C3)=N1)=O
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Chemical Name(2-benzhydryl-5-methyl-1H-imidazole-4-carbonyl)-L-arginine
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Lohman RJ, et al. Nat Commun. 2017 Aug 24;8(1):351.
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