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PI3K-IN-1
CAS No. 1349796-36-6
PI3K-IN-1( SAR245409 | Voxtalisib )
Catalog No. M11414 CAS No. 1349796-36-6
PI3K-IN-1 is a potent inhibitor of PI3K.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 41 | In Stock |
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| 5MG | 65 | In Stock |
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| 10MG | 111 | In Stock |
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| 25MG | 219 | In Stock |
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| 50MG | 305 | In Stock |
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| 100MG | 494 | In Stock |
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| 200MG | Get Quote | In Stock |
|
| 500MG | 1097 | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NamePI3K-IN-1
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NoteResearch use only, not for human use.
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Brief DescriptionPI3K-IN-1 is a potent inhibitor of PI3K.
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DescriptionPI3K-IN-1 is a potent inhibitor of PI3K, extracted from patent WO2012103524 A2 and WO2013147649 A2.(In Vitro):PI3K-IN-1 (25 μM) blocks PI3K/Akt signaling pathways. By using the PI3K inhibitor PI3K-IN-1, TGF-β1 induced transformation into myofibroblast is also inhibited, with relatively reduced expressions of α-SMA, Col-1 and Timp-1.
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In VitroPI3K-IN-1 (25 μM) blocks PI3K/Akt signaling pathways. By using the PI3K inhibitor PI3K-IN-1, TGF-β1 induced transformation into myofibroblast is also inhibited, with relatively reduced expressions of α-SMA, Col-1 and Timp-1.
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In Vivo——
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SynonymsSAR245409 | Voxtalisib
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorDNA-PK|PI3Kα|PI3Kβ|PI3Kγ|PI3Kδ
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1349796-36-6
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Formula Weight599.6569
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Molecular FormulaC31H29N5O6S
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Purity>98% (HPLC)
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SolubilityDMSO: 27.5 mg/mL
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SMILESO=C(NC1=CC=C(S(=O)(NC2=NC3=CC=CC=C3N=C2NC4=CC(OC)=CC(OC)=C4)=O)C=C1)C5=CC=C(C)C(OC)=C5
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Chemical NameN-(4-(N-(3-((3,5-dimethoxyphenyl)amino)quinoxalin-2-yl)sulfamoyl)phenyl)-3-methoxy-4-methylbenzamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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