Endoxifen
CAS No. 112093-28-4
Endoxifen( —— )
Catalog No. M10432 CAS No. 112093-28-4
A metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 69 | In Stock |
|
| 5MG | 61 | In Stock |
|
| 10MG | 81 | In Stock |
|
| 25MG | 170 | In Stock |
|
| 50MG | 268 | In Stock |
|
| 100MG | 402 | In Stock |
|
| 200MG | 582 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
-
Product NameEndoxifen
-
NoteResearch use only, not for human use.
-
Brief DescriptionA metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.
-
DescriptionA metabolite of tamoxifen, orally active non-steroidal selective estrogen receptor modulator (SERM) for the treatment of estrogen receptor-positive breast cancer.Breast Cancer Phase 1 Clinical.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayEndocrinology/Hormones
-
TargetEstrogen Receptor/ERR
-
RecptorER|ERR|hERGPotassiumChannel
-
Research AreaCancer
-
IndicationBreast Cancer
Chemical Information
-
CAS Number112093-28-4
-
Formula Weight373.4874
-
Molecular FormulaC25H27NO2
-
Purity>98% (HPLC)
-
Solubility10 mM in DMSO
-
SMILESCCC(=C(C1=CC=C(C=C1)O)C2=CC=C(C=C2)OCCNC)C3=CC=CC=C3
-
Chemical NamePhenol, 4-[(1Z)-1-[4-[2-(methylamino)ethoxy]phenyl]-2-phenyl-1-buten-1-yl]-
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Brauch H, et al. Clin Chem. 2009 Oct;55(10):1770-82.
2. Markopoulos C, et al. World J Clin Oncol. 2014 Aug 10;5(3):374-81.
3. Mugundu GM, et al. Drug Metab Dispos. 2012 Feb;40(2):389-96.
molnova catalog
related products
-
Estriol
Estriol is an antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast Y cells.
-
Diptoindonesin G
A natural compound, novel chemical probe reciprocally stabilizes ERβ and destabilizes ERα in breast cancer cells.
-
Elacestrant
Elacestrant (RAD-1901) is a novel, orally bioavailable small-molecule selective estrogen receptor degrader (SERD).
Cart
sales@molnova.com