PV-1115

CAS No. 1093793-10-2

PV-1115( PV 1115 | PV1115 )

Catalog No. M10360 CAS No. 1093793-10-2

A potent and highly selective Chk2 inhibitor with IC50 of 0.14 nM; displays greater than 100 uM for Chk1 in vitro.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    PV-1115
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent and highly selective Chk2 inhibitor with IC50 of 0.14 nM; displays greater than 100 uM for Chk1 in vitro.
  • Description
    A potent and highly selective Chk2 inhibitor with IC50 of 0.14 nM; displays greater than 100 uM for Chk1 in vitro.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PV 1115 | PV1115
  • Pathway
    Angiogenesis
  • Target
    Chk
  • Recptor
    Chk
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1093793-10-2
  • Formula Weight
    405.418
  • Molecular Formula
    C20H19N7O3
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    O=C(C(N1)=CC2=C1C([N+]([O-])=O)=CC=C2)NC3=CC=C(/C(C)=N/NC4=NCCN4)C=C3
  • Chemical Name
    N-(4-(1-(2-(4,5-dihydro-1H-imidazol-2-yl)hydrazono)ethyl)phenyl)-7-nitro-1H-indole-2-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Lountos GT, et al. J Struct Biol. 2011 Dec; 176(3):292-301.
molnova catalog
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