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Lys-SMCC-DM1
CAS No. 1281816-04-3
Lys-SMCC-DM1( Lys-Nε-MCC-DM1 )
Catalog No. M23445 CAS No. 1281816-04-3
DM1 is a tubulin inhibitor. Lys-SMCC-DM1 is the active metabolite of DM1.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 1131 | In Stock |
|
| 5MG | 656 | In Stock |
|
| 10MG | 947 | In Stock |
|
| 25MG | 1406 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameLys-SMCC-DM1
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NoteResearch use only, not for human use.
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Brief DescriptionDM1 is a tubulin inhibitor. Lys-SMCC-DM1 is the active metabolite of DM1.
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DescriptionDM1 is a tubulin inhibitor. Lys-SMCC-DM1 is the active metabolite of DM1.
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In Vitro——
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In Vivo——
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SynonymsLys-Nε-MCC-DM1
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetMicrotubule/Tubulin
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Recptortubulin
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Research Area——
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Indication——
Chemical Information
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CAS Number1281816-04-3
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Formula Weight1103.71
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Molecular FormulaC53H75ClN6O15S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (90.60 mM)
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SMILESC[C@@H]1[C@@H]2C[C@]([C@@H](/C=C/C=C(/CC3=CC(=C(C(=C3)OC)Cl)N(C(=O)C[C@@H]([C@]4([C@H]1O4)C)OC(=O)[C@H](C)N(C)C(=O)CCSC5CC(=O)N(C5=O)CC6CCC(CC6)C(=O)NCCCC[C@@H](C(=O)O)N)C)\C)OC)(NC(=O)O2)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Ogitani Y, et al. Bystander killing effect of DS-8201a, a novel anti-human epidermal growth factor receptor 2 antibody-drug conjugate, in tumors with human epidermal growth factor receptor 2 heterogeneity. Cancer Sci. 2016 Jul;107(7):1039-46.
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