KX1-004

CAS No. 518058-84-9

KX1-004( KX1004 | KX 1004 | KX1-004 )

Catalog No. M14808 CAS No. 518058-84-9

KX1-004 is a potent small molecule inhibitor of Src-PTK as a potential protective drug for NIHL.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 49 In Stock
5MG 80 In Stock
10MG 147 In Stock
25MG 267 In Stock
50MG 441 In Stock
100MG 621 In Stock
500MG 1305 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    KX1-004
  • Note
    Research use only, not for human use.
  • Brief Description
    KX1-004 is a potent small molecule inhibitor of Src-PTK as a potential protective drug for NIHL.
  • Description
    KX1-004 is a potent small molecule inhibitor of Src-PTK as a potential protective drug for NIHL.
  • In Vitro
    ——
  • In Vivo
    KX1-004 (30 μM) provides significant protection against noise-induced temporary threshold shift (TTS), permanent threshold shift (PTS) and outer hair cells (OHC) loss.KX1-004 (50 mg/kg) is effective against noise exposure.
  • Synonyms
    KX1004 | KX 1004 | KX1-004
  • Pathway
    Tyrosine Kinase
  • Target
    Src
  • Recptor
    Src-PTK
  • Research Area
    Other Indications
  • Indication
    ——

Chemical Information

  • CAS Number
    518058-84-9
  • Formula Weight
    284.29
  • Molecular Formula
    C16H13FN2O2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: 10 mM
  • SMILES
    O=C(C(N1)=CC2=C1C=CC(F)=C2)NCC3=CC=CC(O)=C3
  • Chemical Name
    5-fluoro-N-(3-hydroxybenzyl)-1H-indole-2-carboxamide.

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Harris KC, et al. Hear Res. 2005 Oct;208(1-2):14-25.
molnova catalog
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