JNJ0966

CAS No. 315705-75-0

JNJ0966( JNJ-0966 | JNJ 0966 | JNJ0966 )

Catalog No. M19325 CAS No. 315705-75-0

JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 68 In Stock
5MG 87 In Stock
10MG 132 In Stock
25MG 290 In Stock
50MG 520 In Stock
100MG 750 In Stock
500MG 1521 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    JNJ0966
  • Note
    Research use only, not for human use.
  • Brief Description
    JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).
  • Description
    JNJ0966 is a highly selective allosteric inhibitor of matrix metalloproteinase-9 (MMP-9).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    JNJ-0966 | JNJ 0966 | JNJ0966
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    P450
  • Recptor
    MMP-9
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    315705-75-0
  • Formula Weight
    360.45
  • Molecular Formula
    C16H16N4O2S2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : 100 mg/mL 277.43 mM; H2O : < 0.1 mg/mL
  • SMILES
    CC1=C(SC(=N1)NC(=O)C)C2=CSC(=N2)NC3=CC=CC=C3OC
  • Chemical Name
    N-(2-((2-Methoxyphenyl)amino)-4'-methyl-[4,5'-bithiazol]-2'-yl)acetamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Scannevin RH, et al. J Biol Chem. 2017 Oct 27;292(43):17963-17974.
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