
ERAP1-IN-1
CAS No. 865273-97-8
ERAP1-IN-1( —— )
Catalog No. M26205 CAS No. 865273-97-8
ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
5MG | 260 | Get Quote |
![]() ![]() |
10MG | 430 | Get Quote |
![]() ![]() |
25MG | 710 | Get Quote |
![]() ![]() |
50MG | 972 | Get Quote |
![]() ![]() |
100MG | 1332 | Get Quote |
![]() ![]() |
500MG | 2673 | Get Quote |
![]() ![]() |
1G | Get Quote | Get Quote |
![]() ![]() |
Biological Information
-
Product NameERAP1-IN-1
-
NoteResearch use only, not for human use.
-
Brief DescriptionERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates.
-
DescriptionERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 competitively inhibits ERAP1 activity towards a nonamer peptide representative of physiological substrates.(In Vitro):ERAP1-IN-1 (50 μM) exhibits specific inhibition of ERAP1 in the cellular context. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayOthers
-
TargetOther Targets
-
RecptorAndrogen Receptor
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number865273-97-8
-
Formula Weight458.45
-
Molecular FormulaC20H21F3N2O5S
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 250 mg/mL (545.32 mM)
-
SMILESCOc1ccc(cc1S(=O)(=O)Nc1cc(ccc1N1CCCCC1)C(F)(F)F)C(O)=O
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1.Coss CC, Bauler M, Narayanan R, Miller DD, Dalton JT. Alanine aminotransferase regulation by androgens in non-hepatic tissues. Pharm Res. 2012 Apr;29(4):1046-56.
molnova catalog



related products
-
Pelgifatamab
Pelgifatamab (BAY-2315497) is a prostate-specific membrane antigen (PSMA) antibody with potential anticancer activity that can be used to study prostate cancer.
-
5(6)-FAM SE
5(6)-FAM SE is an amine-reactive green fluorescent dye widely used for labeling proteins or other molecules that contain a primary or secondary aliphatic amine.
-
4-Bromo-2-(2,6-dioxo...
4-Bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione is a chemical compound.