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CX815
CAS No. 109628-27-5
CX815( CX-815 | CX 815 | NSC 120213 )
Catalog No. M10374 CAS No. 109628-27-5
A novel potent, selective CXCR2 inhibitor with IC50 of 0.4 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
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Biological Information
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Product NameCX815
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NoteResearch use only, not for human use.
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Brief DescriptionA novel potent, selective CXCR2 inhibitor with IC50 of 0.4 nM.
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DescriptionA novel potent, selective CXCR2 inhibitor with IC50 of 0.4 nM; displays>1,000-fold selectivity over CXCR4 (IC50>50 uM); inhibits cell proliferation of H1299 and H460 cells with IC50 of 3.5 and 4.1 uM in MTT assays.
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In Vitro——
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In Vivo——
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SynonymsCX-815 | CX 815 | NSC 120213
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PathwayGPCR/G Protein
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TargetChemokine Receptor
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RecptorChemokine Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number109628-27-5
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Formula Weight327.398
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Molecular FormulaC18H17NO3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : ≥ 100 mg/mL (304.52 mM)
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SMILESCC1=CC=C(C=C1)S(=O)(=O)NC2=C3C(=CC(=C2)OC)C=CC=N3
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Chemical NameN-(6-methoxyquinolin-8-yl)-4-methylbenzenesulfonamide
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Ha H, et al. J Chem Inf Model. 2015 Aug 24;55(8):1720-38.
molnova catalog
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