PCSK9-IN-10

PCSK9-IN-10

Catalog No. M36396

PCSK9-IN-10, a potent and orally active inhibitor of Proprotein Convertase Subtilisin/Kexin Type 9 (PCSK9), exhibits a half-maximal inhibitory concentration (IC50) of 6.4 μM.

Size Price / USD Stock Quantity
2MG 62 Get Quote
5MG 92 Get Quote
10MG 147 Get Quote
25MG 288 Get Quote
50MG 454 Get Quote
100MG 653 Get Quote
500MG 1368 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    PCSK9-IN-10
  • Brief Description
  • Description
  • Storage
  • Note
    Research use only, not for human use.
  • Reference
    1. Qiao MQ, et al. Structure-activity relationship and biological evaluation of xanthine derivatives as PCSK9 inhibitors for the treatment of atherosclerosis. Eur J Med Chem. 2022 Dec 26;247:115047.?
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