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Vafidemstat
CAS No. 1357362-02-7
Vafidemstat( ORY 2001 | ORY-2001 | ORY2001 | Vafidemstat )
Catalog No. M11465 CAS No. 1357362-02-7
Vafidemstat is a novel potent, selective lysine-specific histone demethylase (LSD1) inhibitor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 410 | Get Quote |
|
| 50MG | 1449 | Get Quote |
|
| 100MG | 2196 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameVafidemstat
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NoteResearch use only, not for human use.
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Brief DescriptionVafidemstat is a novel potent, selective lysine-specific histone demethylase (LSD1) inhibitor.
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DescriptionVafidemstat is a novel potent, selective lysine-specific histone demethylase (LSD1) inhibitor.
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In VitroVafidemstat (ORY-2001), a dual LSD1/MAO-B inhibitor, is a novel epigenetic agent for the treatment of neurodegenerative diseases. LSD1 is a protein that participates in transcription regulation complexes; its modulation can be used to tweak transcriptional imbalances in neurodegenerative disease and redress neuroinflammation and cognitive deficit. Vafidemstat (ORY-2001) can be used in the treatment of Alzheimer's disease.
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In Vivo——
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SynonymsORY 2001 | ORY-2001 | ORY2001 | Vafidemstat
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PathwayChromatin/Epigenetic
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TargetHistone Demethylase
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RecptorHistone Demethylase
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Research Area——
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Indication——
Chemical Information
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CAS Number1357362-02-7
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Formula Weight336.395
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Molecular FormulaC19H20N4O2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (148.64 mM)
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SMILES[H][C@@]1([C@@](NCC2=NN=C(N)O2)([H])C1)C(C=C3)=CC=C3OCC4=CC=CC=C4
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Chemical Name1,3,4-Oxadiazole-2-methanamine, 5-amino-N-[(1R,2S)-2-[4-(phenylmethoxy)phenyl]cyclopropyl]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
molnova catalog
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