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Takeda103A

CAS No. 865609-72-9

Takeda103A( Takeda-103-A | Takeda 103 A | Takeda-103A | CMPD103A | CMPD-103A )

Catalog No. M24868 CAS No. 865609-72-9

Takeda103A is the GRK2-dependent bovine tubulin oxidation effective inhibitor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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10MG 406 In Stock
25MG 669 In Stock
50MG 945 In Stock
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Biological Information

  • Product Name
    Takeda103A
  • Note
    Research use only, not for human use.
  • Brief Description
    Takeda103A is the GRK2-dependent bovine tubulin oxidation effective inhibitor.
  • Description
    Takeda103A is the GRK2-dependent bovine tubulin oxidation effective inhibitor.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Takeda-103-A | Takeda 103 A | Takeda-103A | CMPD103A | CMPD-103A
  • Pathway
    Others
  • Target
    GRK (GPCRK)
  • Recptor
    GRK2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    865609-72-9
  • Formula Weight
    463.49
  • Molecular Formula
    C24H23F2N7O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:10 mM
  • SMILES
    CCCN1C(=NN=C1C2=NC=NC=C2)CNC3=CC=CC(=C3)C(=O)NCC4=C(C=CC=C4F)F
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Waldschmidt HV, Homan KT, Cruz-Rodríguez O, et al. Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors. J Med Chem. 2016 Apr 28;59(8):3793-807. doi: 10.1021/acs.jmedchem.5b02000. Epub 2016 Apr 13. PubMed PMID: 27050625.
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