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Serlopitant
CAS No. 860642-69-9
Serlopitant( VPD-737 | MK-0594 )
Catalog No. M16236 CAS No. 860642-69-9
Serlopitant (VPD-737, MK-0594) is a potent, selective substance P/neurokinin 1 (NK1) receptor for treating chronic pruritus.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 1229 | In Stock |
|
| 50MG | 2507 | In Stock |
|
| 100MG | 3168 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSerlopitant
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NoteResearch use only, not for human use.
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Brief DescriptionSerlopitant (VPD-737, MK-0594) is a potent, selective substance P/neurokinin 1 (NK1) receptor for treating chronic pruritus.
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DescriptionSerlopitant (VPD-737, MK-0594) is a potent, selective substance P/neurokinin 1 (NK1) receptor for treating chronic pruritus.Alcoholism Discontinued.
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In Vitro——
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In Vivo——
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SynonymsVPD-737 | MK-0594
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PathwayGPCR/G Protein
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TargetNeurokinin Receptor
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RecptorNeurokinin Receptor
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Research AreaNeurological Disease
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IndicationAlcoholism
Chemical Information
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CAS Number860642-69-9
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Formula Weight555.537
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Molecular FormulaC29H28F7NO2
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C1C=C(N2C[C@@]3([H])CC[C@H](O[C@@H](C4=CC(C(F)(F)F)=CC(C(F)(F)F)=C4)C)[C@@H](C5=CC=C(F)C=C5)[C@]3([H])C2)CC1
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Chemical Name3-((3aR,4R,5S,7aS)-5-((1R)-1-(3,5-bis(Trifluoromethyl)phenyl)ethoxy)-4-(4 fluorophenyl)octahydro-2H-isoindol-2-yl)cyclopent-2-en-1-one
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Yosipovitch G, et al. J Am Acad Dermatol. 2018 May;78(5):882-891.e10.
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