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SJ995973
CAS No. 2882065-25-8
SJ995973( —— )
Catalog No. M37131 CAS No. 2882065-25-8
SJ995973 is a highly potent bromodomain and extraterminal (BET) protein degrader and a BET PROTAC with potential anticancer activity.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 347 | In Stock |
|
| 5MG | 655 | In Stock |
|
| 10MG | 1121 | In Stock |
|
| 25MG | 1638 | In Stock |
|
| 50MG | 2190 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameSJ995973
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NoteResearch use only, not for human use.
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Brief DescriptionSJ995973 is a highly potent bromodomain and extraterminal (BET) protein degrader and a BET PROTAC with potential anticancer activity.
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DescriptionSJ995973 (PROTAC) is a uniquely potent degrader ofbromodomain and extra-terminal (BET) proteins.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorPROTACs
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Research Area——
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Indication——
Chemical Information
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CAS Number2882065-25-8
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Formula Weight730.28
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Molecular FormulaC37H40ClN7O5S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (136.93 mM; Ultrasonic )
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SMILESCC=1C2=C(N3C([C@H](CC(NCCCCCNC(COC4=CC=C(C=C4)C5C(=O)NC(=O)CC5)=O)=O)N=C2C6=CC=C(Cl)C=C6)=NN=C3C)SC1C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Min J, et al. Phenyl-Glutarimides: Alternative Cereblon Binders for the Design of PROTACs. Angew Chem Int Ed Engl. 2021 Dec 13;60(51):26663-26670. ?
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