
RO5166017
CAS No. 1048346-74-2
RO5166017( —— )
Catalog No. M34696 CAS No. 1048346-74-2
RO5166017 is an orally active, potent and selective trace amine-associated receptor 1 (TAAR1) agonist for the study of conditioned taste aversion frontal nerve disorders.
Purity : >98% (HPLC)






Size | Price / USD | Stock | Quantity |
2MG | 141 | Get Quote |
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5MG | 217 | Get Quote |
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10MG | 345 | Get Quote |
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25MG | 569 | Get Quote |
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50MG | 799 | Get Quote |
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100MG | 1017 | Get Quote |
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500MG | Get Quote | Get Quote |
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1G | Get Quote | Get Quote |
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Biological Information
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Product NameRO5166017
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NoteResearch use only, not for human use.
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Brief DescriptionRO5166017 is an orally active, potent and selective trace amine-associated receptor 1 (TAAR1) agonist for the study of conditioned taste aversion frontal nerve disorders.
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DescriptionRO5166017 is an orally active and species-crosses TAAR1 agonist, with Ki values of 1.9 nM, 2.7 nM, 31 nM and 24 nM for mouse, rat, human and cynomolgus monkey, respectively.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorOthers
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Research Area——
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Indication——
Chemical Information
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CAS Number1048346-74-2
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Formula Weight219.28
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Molecular FormulaC12H17N3O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 25 mg/mL (114.01 mM; Ultrasonic )
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SMILESCCN(C[C@H]1COC(N)=N1)c1ccccc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Florent G Revel, et al. TAAR1 activation modulates monoaminergic neurotransmission, preventing hyperdopaminergic and hypoglutamatergic activity. Proc Natl Acad Sci U S A?
molnova catalog



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