Cart
sales@molnova.com
PKC-IN-7
CAS No. 860468-10-6
PKC-IN-7( —— )
Catalog No. M16235 CAS No. 860468-10-6
PKC-IN-7 is a potent, selective, reversible, ATP-competitive PKCα/β inhibitor with IC50 of 4.7/3.3 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 100MG | Get Quote | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NamePKC-IN-7
-
NoteResearch use only, not for human use.
-
Brief DescriptionPKC-IN-7 is a potent, selective, reversible, ATP-competitive PKCα/β inhibitor with IC50 of 4.7/3.3 nM.
-
DescriptionPKC-IN-7 is a potent, selective, reversible, ATP-competitive PKCα/β inhibitor with IC50 of 4.7/3.3 nM; dispalys >50-fold selectivity against PKC isotypes δ,ε,η,θ and other kinases belonging to the AGC family; inhibits IgM-stimulated mouse B cell proliferation with an IC50 of 296 nM.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayAngiogenesis
-
TargetPKC
-
RecptorPKC
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number860468-10-6
-
Formula Weight443.931
-
Molecular FormulaC26H22ClN3O2
-
Purity>98% (HPLC)
-
Solubility——
-
SMILES——
-
Chemical Name3-(2-chloro-7-((dimethylamino)methyl)naphthalen-1-yl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. van Eis MJ, et al. Bioorg Med Chem Lett. 2017 Feb 15;27(4):781-786.
molnova catalog
related products
-
BJE6-106
BJE6-106 (B106)?is a potent, selective PKCδ inhibitor with IC50 of 50 nM, displays excellent selectivity over classical PKC isozymes.
-
CGP60474
A potent CDK1 inhibitor with IC50 of 17 nM; exhibits lower potency at CDK2 and moderate potency at CDK4.
-
Dequalinium chloride
Dequalinium Chloride is a selective blocker of apamin-sensitive K+ channels.
