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PI3Kα-IN-243
CAS No. 1235449-52-1
PI3Kα-IN-243( PI3Kα inhibitor 1 | MDK 9521 | PI3Kα-IN-243 )
Catalog No. M10945 CAS No. 1235449-52-1
A potent PI3Kα inhibitor with IC50 of <0.1 uM; also inhibits HDAC (IC50=0.1-1 uM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 158 | Get Quote |
|
| 5MG | 237 | Get Quote |
|
| 10MG | 357 | Get Quote |
|
| 25MG | 597 | Get Quote |
|
| 50MG | 851 | Get Quote |
|
| 100MG | 1152 | Get Quote |
|
| 500MG | 2313 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePI3Kα-IN-243
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NoteResearch use only, not for human use.
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Brief DescriptionA potent PI3Kα inhibitor with IC50 of <0.1 uM; also inhibits HDAC (IC50=0.1-1 uM).
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DescriptionA potent PI3Kα inhibitor with IC50 of <0.1 uM; also inhibits HDAC (IC50=0.1-1 uM); compound 243 in patent US/20120088764A1.
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In Vitro——
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In Vivo——
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SynonymsPI3Kα inhibitor 1 | MDK 9521 | PI3Kα-IN-243
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorPI3K
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Research AreaCancer
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Indication——
Chemical Information
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CAS Number1235449-52-1
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Formula Weight507.5681
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Molecular FormulaC23H25N9O3S
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Purity>98% (HPLC)
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SolubilityDMSO: ≥ 37 mg/mL
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SMILESO=C(C1=CN=C(N(C)CC2=CC3=NC(C4=CC=C(NC)N=C4)=NC(N5CCOCC5)=C3S2)N=C1)NO
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Chemical Name5-Pyrimidinecarboxamide, N-hydroxy-2-[methyl[[2-[6-(methylamino)-3-pyridinyl]-4-(4-morpholinyl)thieno[3,2-d]pyrimidin-6-yl]methyl]amino]-
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Patent US/20120088764A1
molnova catalog
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