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Home - Products - GPCR/G Protein - Glucagon Receptor - PF-06882961

PF-06882961

CAS No. 2230198-02-2

PF-06882961( —— )

Catalog No. M22917 CAS No. 2230198-02-2

PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist. PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat.

Purity : >98% (HPLC)

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Biological Information

  • Product Name
    PF-06882961
  • Note
    Research use only, not for human use.
  • Brief Description
    PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist. PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat.
  • Description
    PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist. PF-06882961 shows mild to moderate damage to the heart, moderate to severe effects on the thymus gland (which helps with managing infection), mild to moderate stomach ulcers at the highest dose level given in the rat.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Glucagon Receptor
  • Recptor
    GLP-1
  • Research Area
    Metabolism
  • Indication
    Diabetes Mellitus, Type 2

Chemical Information

  • CAS Number
    2230198-02-2
  • Formula Weight
    555.6
  • Molecular Formula
    C31H30FN5O4
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:125 mg/mL (224.98 mM; Need ultrasonic)
  • SMILES
    OC(C1=CC=C(N=C(CN2CCC(C3=NC(OCC4=CC=C(C#N)C=C4F)=CC=C3)CC2)N5C[C@H]6OCC6)C5=C1)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. 20th SCI/RSC Medicinal Chemistry Symposium.
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