Cart
sales@molnova.com
NPAS3-IN-1
CAS No. 2207-44-5
NPAS3-IN-1( —— )
Catalog No. M37303 CAS No. 2207-44-5
NPAS3-IN-1 is a potent inhibitor of NPAS3-ARNT heterodimerization, modulating NPAS3 transcription by targeting the interaction between NPAS3 and ARNT at the cellular level.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 116 | Get Quote |
|
| 5MG | 179 | Get Quote |
|
| 10MG | 282 | Get Quote |
|
| 25MG | 477 | Get Quote |
|
| 50MG | 679 | Get Quote |
|
| 100MG | 888 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
-
Product NameNPAS3-IN-1
-
NoteResearch use only, not for human use.
-
Brief DescriptionNPAS3-IN-1 is a potent inhibitor of NPAS3-ARNT heterodimerization, modulating NPAS3 transcription by targeting the interaction between NPAS3 and ARNT at the cellular level.
-
DescriptionNPAS3-IN-1 is a potent inhibitor of NPAS3-ARNT heterodimerization and regulates NPAS3 transcription by disrupting the heterodimerization of NPAS3 with ARNT at the cellular level.
-
In Vitro——
-
In Vivo——
-
Synonyms——
-
PathwayOthers
-
TargetOther Targets
-
RecptorOthers
-
Research Area——
-
Indication——
Chemical Information
-
CAS Number2207-44-5
-
Formula Weight295.36
-
Molecular FormulaC10H5N3O2S3
-
Purity>98% (HPLC)
-
SolubilityIn Vitro:?DMSO : 25 mg/mL (84.64 mM; Ultrasonic )
-
SMILESO=[N+]([O-])C1=CN=C(SC2=NC3=C(S2)C=CC=C3)S1
-
Chemical Name——
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Li P, et al. Discovery of a highly potent NPAS3 heterodimer inhibitor by covalently modifying ARNT. Bioorg Chem. 2023 Oct;139:106676.?
molnova catalog
related products
-
[Phe1Ψ(CH2-NH)Gly2]N...
Potent agonist of the nociceptin (ORL1) receptor, demonstrated both in vitro and in vivo. Selective, competitive antagonism at the nociceptin receptor has also been reported (pA2 = 7.02 and 6.75 in the guinea pig ileum and mouse vas deferens respectively).
-
2,4-Dihydroxydihydro...
2',4'-Dihydroxydihydrochalcone has cytotoxic, and anti-inflammatory activities.
-
NH2-C5-NH-Boc
NH2-C5-NH-Boc (PROTAC Linker 23) is an alkyl chain-based PROTAC linker that can be used in the synthesis of PROTACs.
