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GLPG3970
CAS No. 2403733-82-2
GLPG3970( —— )
Catalog No. M36521 CAS No. 2403733-82-2
GLPG3970 GLPG3970 is a novel orally available selective dual SIK2/SIK3 inhibitor.GLPG3970 has potential anti-inflammatory activity for the study of autoimmune diseases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 150 | In Stock |
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| 5MG | 132 | In Stock |
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| 10MG | 188 | In Stock |
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| 25MG | 395 | In Stock |
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| 50MG | 581 | In Stock |
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| 100MG | 828 | In Stock |
|
| 200MG | 1135 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGLPG3970
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NoteResearch use only, not for human use.
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Brief DescriptionGLPG3970 GLPG3970 is a novel orally available selective dual SIK2/SIK3 inhibitor.GLPG3970 has potential anti-inflammatory activity for the study of autoimmune diseases.
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DescriptionGLPG3970 (compound 88) is a first-in-class SIK2/SIK3 inhibitor. GLPG3970 can be used for the research of inflammation and autoimmune disease.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayAutophagy
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TargetSIK
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RecptorSIK
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Research Area——
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Indication——
Chemical Information
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CAS Number2403733-82-2
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Formula Weight504.5
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Molecular FormulaC25H27F3N4O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (198.22 mM; Ultrasonic )
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SMILESO=C1C=2C(OC)=CC(=CC2CCN1CC(F)(F)F)C3=CN=C4C=C(OCCN5CCOCC5)C=CN43
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. DESROY N, et al. NOVEL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF DISEASES. WO/2019/238424. 2019.
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