RORγ inverse agonist 1

CAS No. 529500-72-9

RORγ inverse agonist 1( —— )

Catalog No. M36101 CAS No. 529500-72-9

RORγ inverse agonist 1 has anti-inflammatory activity and can be used to treat rheumatism and psoriasis.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 45 In Stock
10MG 72 In Stock
25MG 116 In Stock
50MG 172 In Stock
100MG 250 In Stock
500MG 609 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    RORγ inverse agonist 1
  • Note
    Research use only, not for human use.
  • Brief Description
    RORγ inverse agonist 1 has anti-inflammatory activity and can be used to treat rheumatism and psoriasis.
  • Description
    RORγ inverse agonist 1 is the inverse agonist of RORγ.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    Others
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    529500-72-9
  • Formula Weight
    463.47
  • Molecular Formula
    C22H20F3N3O3S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    N(S(=O)(=O)C1=CC=C(C)C=C1)(CC(NCC=2C=CN=CC2)=O)C3=CC(C(F)(F)F)=CC=C3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Song Y, et al. Identification of N-phenyl-2-(N-phenylphenylsulfonamido)acetamides as new RORγ inverse agonists: Virtual screening, structure-based optimization, and biological evaluation. Eur J Med Chem. 2016 Jun 30;116:13-26.?
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