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BJJF078
CAS No. 2531244-56-9
BJJF078( —— )
Catalog No. M36035 CAS No. 2531244-56-9
BJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 and 54 nM for human and mouse glutamine aminotransferase, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 103 | In Stock |
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| 10MG | 145 | In Stock |
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| 25MG | 250 | In Stock |
|
| 50MG | 365 | In Stock |
|
| 100MG | 538 | In Stock |
|
| 200MG | 768 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBJJF078
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NoteResearch use only, not for human use.
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Brief DescriptionBJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 and 54 nM for human and mouse glutamine aminotransferase, respectively.
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DescriptionBJJF078 is an aminopiperidine derivative. BJJF078 is a potent inhibitor of recombinant human and mouse Transglutaminase enzyme (TG2) activity, IC50 values of 41 and 54 nM, respectively. BJJF078 also inhibits the close related enzyme TG1, with an IC50 of 0.16 μM. BJJF078 can be used for Multiple sclerosis (MS) research.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorGlutaminase
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Research Area——
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Indication——
Chemical Information
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CAS Number2531244-56-9
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Formula Weight523.6
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Molecular FormulaC27H29N3O6S
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Purity>98% (HPLC)
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Solubility——
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SMILESS(=O)(=O)(C=1C2=C(C(NC(=O)C3=CC(OC)=C(OC)C=C3)=CC=C2)C=CC1)N4CCC(NC(C=C)=O)CC4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Chrobok NL, et al. Characterization of Transglutaminase 2 activity inhibitors in monocytes in vitro and their effect in a mouse model for multiple sclerosis. PLoS One. 2018 Apr 24;13(4):e0196433.?
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