Linagliptin Methyldimer

CAS No. 1418133-47-7

Linagliptin Methyldimer( —— )

Catalog No. M36028 CAS No. 1418133-47-7

Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 161 In Stock
5MG 275 In Stock
10MG 407 In Stock
25MG 663 In Stock
50MG 900 In Stock
100MG 1190 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Linagliptin Methyldimer
  • Note
    Research use only, not for human use.
  • Brief Description
    Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.
  • Description
    Linagliptin methyldimer is an impurity of Linagliptin. Linagliptin is a DPP-IV inhibitor, with IC50 of 1 nM.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    Proteasome
  • Recptor
    Proteasome
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1418133-47-7
  • Formula Weight
    945.08
  • Molecular Formula
    C50H56N16O4
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    C(C#CC)N1C2=C(N=C1N3C[C@H](N)CCC3)N(C)C(=O)N(CC4=NC(CC=5C6=C(N=C(CN7C(=O)C=8N(CC#CC)C(=NC8N(C)C7=O)N9C[C@H](N)CCC9)N5)C=CC=C6)(C)C=%10C(N4)=CC=CC%10)C2=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Pfrengle, et al. Substituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions as DPP-IV inhibitors. Patent. WO2013010964 A1.
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