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Linagliptin Methyldimer
CAS No. 1418133-47-7
Linagliptin Methyldimer( —— )
Catalog No. M36028 CAS No. 1418133-47-7
Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 178 | Get Quote |
|
| 5MG | 275 | Get Quote |
|
| 10MG | 407 | Get Quote |
|
| 25MG | 642 | Get Quote |
|
| 50MG | 891 | Get Quote |
|
| 100MG | 1152 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameLinagliptin Methyldimer
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NoteResearch use only, not for human use.
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Brief DescriptionLinagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.
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DescriptionLinagliptin methyldimer is an impurity of Linagliptin. Linagliptin is a DPP-IV inhibitor, with IC50 of 1 nM.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayProteasome/Ubiquitin
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TargetProteasome
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RecptorProteasome
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Research Area——
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Indication——
Chemical Information
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CAS Number1418133-47-7
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Formula Weight945.08
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Molecular FormulaC50H56N16O4
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Purity>98% (HPLC)
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Solubility——
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SMILESC(C#CC)N1C2=C(N=C1N3C[C@H](N)CCC3)N(C)C(=O)N(CC4=NC(CC=5C6=C(N=C(CN7C(=O)C=8N(CC#CC)C(=NC8N(C)C7=O)N9C[C@H](N)CCC9)N5)C=CC=C6)(C)C=%10C(N4)=CC=CC%10)C2=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Pfrengle, et al. Substituted quinazolines, the preparation thereof and the use thereof in pharmaceutical compositions as DPP-IV inhibitors. Patent. WO2013010964 A1.
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