SLK/STK10-IN-1

CAS No. 264210-49-3

SLK/STK10-IN-1( —— )

Catalog No. M35494 CAS No. 264210-49-3

SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    SLK/STK10-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    SLK/STK10-IN-1 is a selective and potent inhibitor of SLK and STK10 with potential antitumor activity.
  • Description
    SLK/STK10-IN-1 is a potent and selective inhibitor of SLK and STK10 with nanomolar potency.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    Serine Protease
  • Recptor
    Serine Protease
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    264210-49-3
  • Formula Weight
    328.75
  • Molecular Formula
    C17H13ClN2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (304.18 mM; Ultrasonic )
  • SMILES
    O=C1NC(=O)C(C=2C=CC=CC2OC)=C1NC=3C=CC=C(Cl)C3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Serafim RAM, et al. Discovery of a Potent Dual SLK/STK10 Inhibitor Based on a Maleimide Scaffold. J Med Chem. 2021 Sep 23;64(18):13259-13278. ?
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