Cathepsin X-IN-1

CAS No. 2418577-51-0

Cathepsin X-IN-1( —— )

Catalog No. M35476 CAS No. 2418577-51-0

Cathepsin X-IN-1 (compound 25) is a potent Cathepsin X inhibitor (IC50 = 7.13 μM) that reduces PC-3 cell migration with low cytotoxicity .

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 33 In Stock
5MG 55 In Stock
10MG 93 In Stock
25MG 187 In Stock
50MG 300 In Stock
100MG 433 In Stock
200MG 603 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Cathepsin X-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    Cathepsin X-IN-1 (compound 25) is a potent Cathepsin X inhibitor (IC50 = 7.13 μM) that reduces PC-3 cell migration with low cytotoxicity .
  • Description
    Cathepsin X-IN-1 (compound 25) is a potent Cathepsin X inhibitor with an IC50 of 7.13 μM. Cathepsin X-IN-1 decreases PC-3 cell migration with low cytotoxic.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    Cysteine Protease
  • Recptor
    Cysteine Protease
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2418577-51-0
  • Formula Weight
    315.35
  • Molecular Formula
    C15H13N3O3S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : ≥ 100 mg/mL (317.11 mM; )H2O : ≥ 4.85 mg/mL (15.38 mM)
  • SMILES
    O=C(CSc1nccn1CC#N)c1ccc2OCCOc2c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Fonovi? UP, et al. Structure-activity relationships of triazole-benzodioxine inhibitors of cathepsin X. Eur J Med Chem. 2020 May 1;193:112218.?
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