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GLP-1R modulator C16

CAS No. 875005-43-9

GLP-1R modulator C16( —— )

Catalog No. M35241 CAS No. 875005-43-9

GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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Biological Information

Product Name

GLP-1R modulator C16
Note

Research use only, not for human use.
Brief Description

GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.
Description

GLP-1R modulator C16 is an allosteric modulator enhancing GLP-1 binding to GLP-1R via a transmembrane site (EC50 8.43 ± 3.82 μM).
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

GPCR/G Protein
Target

Glucagon Receptor
Recptor

Glucagon Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

875005-43-9
Formula Weight

408.89
Molecular Formula

C21H26ClFN2O3
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 50 mg/mL (122.28 mM; Ultrasonic (<60°C)
SMILES

COc1cc(CNCCN2CCOCC2)ccc1OCc1c(F)cccc1Cl
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Wang J, et al. Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site. ACS Chem Biol. 2021 Nov 19;16(11):2444-2452. ?

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