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TIBI
CAS No. 1196457-06-3
TIBI( —— )
Catalog No. M34446 CAS No. 1196457-06-3
TIBI is an ATP-competitive Rio1 inhibitor that acts in a similar manner to fungamycin and enhances the thermal stability of the enzyme.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 50MG | 657 | Get Quote |
|
| 100MG | 1026 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameTIBI
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NoteResearch use only, not for human use.
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Brief DescriptionTIBI is an ATP-competitive Rio1 inhibitor that acts in a similar manner to fungamycin and enhances the thermal stability of the enzyme.
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DescriptionTIBI is a potent and ATP-competitive inhibitor of Rio1 (IC50: 0.09 μM, Ki: 0.05 μM). TIBI enhances the thermostability of the enzyme Rio1.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorOthers
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Research Area——
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Indication——
Chemical Information
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CAS Number1196457-06-3
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Formula Weight621.72
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Molecular FormulaC7H2I4N2
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (80.42 mM; Ultrasonic )
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SMILESIC=1C(I)=C(I)C=2NC=NC2C1I
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kubiński K, et al. Benzimidazole inhibitors of protein kinase CK2 potently inhibit the activity of atypical protein kinase Rio1. Mol Cell Biochem. 2017 Feb;426(1-2):195-203.?
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