BPDBA( —— )

Catalog No. M34193 CAS No. 312281-74-6

BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and mouse GAT2, with IC50 values of 20 μM and 35 μM, respectively.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	44	In Stock
10MG	35	In Stock
25MG	74	In Stock
50MG	116	In Stock
100MG	187	In Stock
200MG	Get Quote	In Stock
500MG	432	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

BPDBA
Note

Research use only, not for human use.
Brief Description

BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and mouse GAT2, with IC50 values of 20 μM and 35 μM, respectively.
Description

BPDBA is a selective and noncompetitive betaine/GABA transporter (BGT-1) inhibitor with IC50s of 20 μM and 35 μM against human BGT-1 and mouse GAT2, respectively.
In Vitro

——
In Vivo

——
Synonyms

——
Pathway

Others
Target

Other Targets
Recptor

GABA Receptor
Research Area

——
Indication

——

Chemical Information

CAS Number

312281-74-6
Formula Weight

363.28
Molecular Formula

C19H20Cl2N2O
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 100 mg/mL (275.27 mM; Ultrasonic )
SMILES

C(N1CCC(NC(=O)C2=C(Cl)C=C(Cl)C=C2)CC1)C3=CC=CC=C3
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1. Kragholm B, et al. Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile. Biochem Pharmacol. 2013 Aug 15;86(4):521-8.?

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