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PI3Kδ-IN-3
CAS No. 1431540-99-6
PI3Kδ-IN-3( —— )
Catalog No. M34137 CAS No. 1431540-99-6
PI3Kδ-IN-3 (TC KHNS 11) is a PI3Kδ inhibitor with an IC50 value of 9 nM.PI3Kδ-IN-3 has a favorable pharmacokinetic profile and inhibits B cell function.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 131 | Get Quote |
|
| 5MG | 185 | Get Quote |
|
| 10MG | 295 | Get Quote |
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| 25MG | 487 | Get Quote |
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| 50MG | 704 | Get Quote |
|
| 100MG | 963 | Get Quote |
|
| 500MG | 1935 | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePI3Kδ-IN-3
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NoteResearch use only, not for human use.
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Brief DescriptionPI3Kδ-IN-3 (TC KHNS 11) is a PI3Kδ inhibitor with an IC50 value of 9 nM.PI3Kδ-IN-3 has a favorable pharmacokinetic profile and inhibits B cell function.
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DescriptionPI3Kδ-IN-3 (Compound 11) is a PI3Kδ inhibitor (IC50: 9 nM). PI3Kδ-IN-3 inhibits B cell function. PI3Kδ-IN-3 has good pharmacokinetic properties.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayPI3K/Akt/mTOR signaling
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TargetPI3K
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RecptorPI3K
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Research Area——
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Indication——
Chemical Information
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CAS Number1431540-99-6
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Formula Weight492.53
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Molecular FormulaC28H24N6O3
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Purity>98% (HPLC)
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Solubility——
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SMILESC(=O)(C=1C=C(C=2C3=C(C=CC(=C3)C=4C=C(C#N)C(OC)=NC4)N=CN2)C=CC1)N5CCN(C(C)=O)CC5
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Hoegenauer K, et al. Discovery and Pharmacological Characterization of Novel Quinazoline-Based PI3K Delta-Selective Inhibitors. ACS Med Chem Lett. 2016 Jun 2;7(8):762-7.?
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