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Rilmakalim
CAS No. 132014-21-2
Rilmakalim( —— )
Catalog No. M34129 CAS No. 132014-21-2
Rilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 304 | In Stock |
|
| 10MG | 456 | In Stock |
|
| 25MG | 747 | In Stock |
|
| 50MG | 1004 | In Stock |
|
| 100MG | Get Quote | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameRilmakalim
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NoteResearch use only, not for human use.
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Brief DescriptionRilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect.
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DescriptionRilmakalim (HOE 234) is a potassium channel opener(PCO) that activates ATP-sensitive K+ channels in theheart or other tissues.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetSodium Channel
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RecptorSodium Channel
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Research Area——
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Indication——
Chemical Information
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CAS Number132014-21-2
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Formula Weight401.48
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Molecular FormulaC21H23NO5S
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Purity>98% (HPLC)
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Solubility——
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SMILESO[C@H]1[C@@H](C=2C(=CC=C(S(=O)(=O)C3=CC=CC=C3)C2)OC1(C)C)N4C(=O)CCC4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Kocic, Ivanet al. Hypotonic stress increases efficacy of rilmakalim, but not pinacidil, toactivate ATP-sensitive K(+) current in guinea pig ventricular myocytes. Journalof pharmacological sciences vol. 95,2 (2004): 189-95.?
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