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GW438014A
CAS No. 469861-49-2
GW438014A( —— )
Catalog No. M33987 CAS No. 469861-49-2
GW438014A is a potent, selective antagonist of the NPY-Y5 receptor, effectively inhibiting food consumption and curbing body weight gain in obese rodents.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 32 | In Stock |
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| 10MG | 51 | In Stock |
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| 25MG | 105 | In Stock |
|
| 50MG | 161 | In Stock |
|
| 100MG | 230 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameGW438014A
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NoteResearch use only, not for human use.
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Brief DescriptionGW438014A is a potent, selective antagonist of the NPY-Y5 receptor, effectively inhibiting food consumption and curbing body weight gain in obese rodents.
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DescriptionGW438014A is a potent and selective NPY-Y5 receptor antagonist. GW438014A inhibits food intake and reduces body weight gain in obese rodents.
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In Vitro——
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In VivoAnimal Model:obese ob/ob mice Dosage:10 mg/kg Administration:intraperitoneal injection; daily, for 7 d Result:Decreased the rate of weight gain in both lean and obese rats.
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Synonyms——
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PathwayGPCR/G Protein
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TargetNeuropeptide Y Receptor
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RecptorNeuropeptide Y Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number469861-49-2
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Formula Weight437.51
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Molecular FormulaC23H23N3O4S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (571.42 mM; Ultrasonic )
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SMILESO=C(NC1=NC=2C=CC=CC2N1CCC=3C=CC=CC3)C=4C=CC=CC4.O=S(=O)(O)C
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Daniels AJ, et, al. Food intake inhibition and reduction in body weight gain in lean and obese rodents treated with GW438014A, a potent and selective NPY-Y5 receptor antagonist. Regul Pept. 2002 Jun 15;106(1-3):47-54.?
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