(±)-AC 7954 hydrochloride

CAS No. 477313-09-0

(±)-AC 7954 hydrochloride( —— )

Catalog No. M33818 CAS No. 477313-09-0

(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 122 In Stock
5MG 113 In Stock
10MG 167 In Stock
25MG 282 In Stock
50MG 403 In Stock
100MG 551 In Stock
200MG 728 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    (±)-AC 7954 hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    (±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.
  • Description
    AC-7954 is a selective nonpeptidic urotensin receptor agonist (EC50: 300 nM at the human UII receptor).
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    GPCR/G Protein
  • Target
    Neurotensin Receptor
  • Recptor
    Neurotensin Receptor
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    477313-09-0
  • Formula Weight
    366.28
  • Molecular Formula
    C19H21Cl2NO2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    Cl.O=C1OC(C2=CC=C(Cl)C=C2)(CC=3C=CC=CC13)CCN(C)C
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Croston GE, et al. Discovery of the first nonpeptide agonist of the GPR14/urotensin-II receptor: 3-(4-chlorophenyl)-3-(2- (dimethylamino)ethyl)isochroman-1-one (AC-7954). J Med Chem. 2002 Nov 7;45(23):4950-3.?
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