αvβ1 integrin-IN-1

CAS No. 1689540-62-2

αvβ1 integrin-IN-1( —— )

Catalog No. M33190 CAS No. 1689540-62-2

αvβ1 integrin-IN-1 is a potent and selective inhibitor of αvβ1 integrin (IC50 of 0.63 nM) with antifibrotic effects.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 337 In Stock
5MG 275 In Stock
10MG 432 In Stock
25MG 696 In Stock
50MG 918 In Stock
100MG 1265 In Stock
200MG 1702 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    αvβ1 integrin-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    αvβ1 integrin-IN-1 is a potent and selective inhibitor of αvβ1 integrin (IC50 of 0.63 nM) with antifibrotic effects.
  • Description
    αvβ1 integrin-IN-1 (Compound C8) is a potent and selective αvβ1 integrin inhibitor with an IC50 of 0.63 nM. Antifibrotic effects.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Integrin
  • Recptor
    Integrin
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1689540-62-2
  • Formula Weight
    558.65
  • Molecular Formula
    C26H34N6O6S
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    S(=O)(=O)(N1[C@H](C(N[C@@H](CC2=CC=C(NC(CCCCNC(=N)N)=O)C=C2)C(O)=O)=O)CCC1)C3=CC=CC=C3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Reed NI, et al. Exploring N-Arylsulfonyl-l-proline Scaffold as a Platform for Potent and Selective αvβ1 Integrin Inhibitors. ACS Med Chem Lett. 2016 Aug 30;7(10):902-907.?
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