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(Rac)-VU 6008667

CAS No. 2092917-63-8

(Rac)-VU 6008667( —— )

Catalog No. M33096 CAS No. 2092917-63-8

(Rac)-VU 6008667 is a selective negative allosteric modulator of the muscarinic acetylcholine receptor subtype 5 (M5 NAM), with an IC50 of 1.8 μM and a pIC50 of 5.75, exhibiting high CNS penetration.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
2MG	32	In Stock
5MG	59	In Stock
10MG	107	In Stock
25MG	183	In Stock
50MG	263	In Stock
100MG	393	In Stock
200MG	548	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

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Biological Information

Product Name

(Rac)-VU 6008667
Note

Research use only, not for human use.
Brief Description

(Rac)-VU 6008667 is a selective negative allosteric modulator of the muscarinic acetylcholine receptor subtype 5 (M5 NAM), with an IC50 of 1.8 μM and a pIC50 of 5.75, exhibiting high CNS penetration.
Description

(Rac)-VU 6008667 is a selective negative allosteric modulator of the muscarinic acetylcholine receptor subtype 5 (M5 NAM), with an IC50 of 1.8 μM and a pIC50 of 5.75, exhibiting high CNS penetration.
In Vitro

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In Vivo

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Synonyms

——
Pathway

Cell Cycle/DNA Damage
Target

AChR
Recptor

AChR
Research Area

——
Indication

——

Chemical Information

CAS Number

2092917-63-8
Formula Weight

438.85
Molecular Formula

C24H17ClF2N2O2
Purity

>98% (HPLC)
Solubility

——
SMILES

C(=O)(N1C2(C=3C(C(=O)N2CC1)=CC=CC3)C4=CC(C)=C(Cl)C=C4)C5=CC(F)=C(F)C=C5
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

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