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NF-56-EJ40 hydrochloride

CAS No. 2728500-80-7

NF-56-EJ40 hydrochloride( —— )

Catalog No. M33038 CAS No. 2728500-80-7

NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1.

Purity : >98% (HPLC)

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Size	Price / USD	Stock	Quantity
5MG	48	Get Quote
10MG	71	Get Quote
25MG	118	Get Quote
50MG	177	Get Quote
100MG	258	Get Quote
200MG	388	Get Quote
500MG	Get Quote	Get Quote
1G	Get Quote	Get Quote

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Biological Information

Product Name

NF-56-EJ40 hydrochloride
Note

Research use only, not for human use.
Brief Description

NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1.
Description

NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 hydrochloride has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM.
In Vitro

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In Vivo

——
Synonyms

——
Pathway

GPCR/G Protein
Target

GHSR
Recptor

GHSR
Research Area

——
Indication

——

Chemical Information

CAS Number

2728500-80-7
Formula Weight

516.46
Molecular Formula

C27H31Cl2N3O3
Purity

>98% (HPLC)
Solubility

——
SMILES

O=C(CC1=C(NC(C2=CC=CC(C3=CC=C(CN4CCN(CC4)C)C=C3)=C2)=O)C=CC=C1)O.Cl.Cl
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

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