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KI696 isomer
CAS No. 1799974-69-8
KI696 isomer( —— )
Catalog No. M32981 CAS No. 1799974-69-8
KI696 isomer is an isomer of KI696, a low affinity probe for the study of immune and metabolic diseases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 306 | In Stock |
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| 5MG | 278 | In Stock |
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| 10MG | 466 | In Stock |
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| 25MG | 941 | In Stock |
|
| 50MG | 1237 | In Stock |
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| 100MG | 1628 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameKI696 isomer
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NoteResearch use only, not for human use.
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Brief DescriptionKI696 isomer is an isomer of KI696, a low affinity probe for the study of immune and metabolic diseases.
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DescriptionKI696 isomer is the less active isomer of KI696 (HY-101140). KI696 is a high affinity probe that disrupts the Keap1/NRF2 interaction.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayNuclear Receptor/Transcription Factor
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TargetKeap1-Nrf2
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RecptorNrf2
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Research Area——
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Indication——
Chemical Information
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CAS Number1799974-69-8
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Formula Weight550.63
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Molecular FormulaC28H30N4O6S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (227.01 mM; Ultrasonic )
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SMILESCOc1cc(cc2nnn(C)c12)[C@H](CC(O)=O)c1ccc(C)c(CN2C[C@@H](C)Oc3ccccc3S2(=O)=O)c1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Davies TG, et al. Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery. J Med Chem. 2016 Apr 28?
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