AHR antagonist 2
CAS No. 2338747-54-7
AHR antagonist 2( —— )
Catalog No. M32773 CAS No. 2338747-54-7
AHR antagonist 2 is an antagonist of the aryl hydrocarbon receptor. The IC50s for human AHR and mouse AHR are 0.885 and 2.03 nM, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 74 | Get Quote |
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| 5MG | 112 | Get Quote |
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| 10MG | 186 | Get Quote |
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| 25MG | 307 | Get Quote |
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| 50MG | 434 | Get Quote |
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| 100MG | 605 | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameAHR antagonist 2
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NoteResearch use only, not for human use.
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Brief DescriptionAHR antagonist 2 is an antagonist of the aryl hydrocarbon receptor. The IC50s for human AHR and mouse AHR are 0.885 and 2.03 nM, respectively.
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DescriptionAHR antagonist 2 is a potent aryl hydrocarbon receptor (AHR) antagonist, extracted from patent WO2019101641A1, compound example 1, with IC50s of 0.885 and 2.03 nM for human and mouse AhR.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorAryl Hydrocarbon Receptor
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Research Area——
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Indication——
Chemical Information
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CAS Number2338747-54-7
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Formula Weight418.37
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Molecular FormulaC20H17F3N4O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 250 mg/mL (597.56 mM; Ultrasonic )
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SMILESC[C@@H](CO)NC(=O)c1cc(nc(n1)-c1cccnc1)-c1ccc(OC(F)(F)F)cc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
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