Cevidoplenib dimesylate hydrochloride
CAS No. 269062-93-3
Cevidoplenib dimesylate hydrochloride( Cevidoplenib dimesylate hydrochloride(2043659-93-2 Free base) )
Catalog No. M28906 CAS No. 269062-93-3
Cevidoplenib dimesylate hydrochloride is a spleen tyrosine kinase (Syk) inhibitor showing potential immunomodulating and anti-inflammatory properties.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 223 | Get Quote |
|
| 10MG | 357 | Get Quote |
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| 25MG | 597 | Get Quote |
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| 50MG | 851 | Get Quote |
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| 100MG | 1152 | Get Quote |
|
| 500MG | 2313 | Get Quote |
|
| 1G | Get Quote | Get Quote |
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Biological Information
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Product NameCevidoplenib dimesylate hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionCevidoplenib dimesylate hydrochloride is a spleen tyrosine kinase (Syk) inhibitor showing potential immunomodulating and anti-inflammatory properties.
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DescriptionCevidoplenib dimesylate hydrochloride is a spleen tyrosine kinase (Syk) inhibitor showing potential immunomodulating and anti-inflammatory properties.(In Vitro):Cevidoplenib dimesylate hydrochloride(oral) inhibited the activity of SYK and blocked Fc receptor and B-cell receptor (BCR)-mediated signaling in inflammatory cells, including macrophages, mast cells, natural killer cells, B cells, and neutrophils.
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In Vitro——
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In Vivo——
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SynonymsCevidoplenib dimesylate hydrochloride(2043659-93-2 Free base)
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PathwayAngiogenesis
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TargetSyk
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RecptorAdenylyl cyclase (AC)
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Research Area——
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Indication——
Chemical Information
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CAS Number269062-93-3
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Formula Weight1957.9
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Molecular FormulaC90H132Cl5N27O12
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Purity>98% (HPLC)
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Solubility——
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SMILESNCCCC[C@@H](C(N)=O)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](CC1=CNC2=C1C=CC=C2)NC([C@H]3N(C([C@H](CC4=CNC5=C4C=CC=C5)NC([C@H](CC6=CNC7=C6C=CC=C7)NC([C@H]8N(C([C@H](CC9=CNC%10=C9C=CC=C%10)NC([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@H]([C@@H](C)CC)N)=
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Ramos-Espiritu L, et al. Discovery of LRE1 as a specific and allosteric inhibitor of soluble adenylyl cyclase. Nat Chem Biol. 2016 Oct;12(10):838-44.
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