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Eclitasertib
CAS No. 2125450-76-0
Eclitasertib( DNL-758 | SAR-443122 )
Catalog No. M28842 CAS No. 2125450-76-0
Eclitasertib is a potent inhibitor of receptor-interacting protein kinase 1 (RIPK1, IC50 of <1 μΜ).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 250 | In Stock |
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| 2MG | 145 | In Stock |
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| 5MG | 227 | In Stock |
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| 10MG | 359 | In Stock |
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| 25MG | 653 | In Stock |
|
| 50MG | 886 | In Stock |
|
| 100MG | 1265 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameEclitasertib
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NoteResearch use only, not for human use.
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Brief DescriptionEclitasertib is a potent inhibitor of receptor-interacting protein kinase 1 (RIPK1, IC50 of <1 μΜ).
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DescriptionEclitasertib is a potent inhibitor of receptor-interacting protein kinase 1 (RIPK1, IC50 of <1 μΜ).
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In Vitro——
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In Vivo——
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SynonymsDNL-758 | SAR-443122
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PathwayApoptosis
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TargetRIP kinase
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RecptorGLUT
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Research Area——
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Indication——
Chemical Information
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CAS Number2125450-76-0
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Formula Weight378.38
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Molecular FormulaC19H18N6O3
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (330.36 mM)
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SMILESCN(c1ncccc1OC[C@@H]1NC(c2nc(Cc3ccccc3)n[nH]2)=O)C1=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Liu KG, et al. Discovery and Optimization of Glucose Uptake Inhibitors. J Med Chem. 2020;63(10):5201-5211.
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