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(E)-Akt inhibitor-IV
CAS No. 959841-49-7
(E)-Akt inhibitor-IV( (E)-Akt inhibitor-IV? | CS-1992 | (E)-AKTIV )
Catalog No. M28654 CAS No. 959841-49-7
(E)-Akt inhibitor-IV ((E)-AKTIV) is an inhibitor of PI3K-Akt.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 151 | In Stock |
|
| 5MG | 112 | In Stock |
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| 10MG | 180 | In Stock |
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| 25MG | 337 | In Stock |
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| 50MG | 458 | In Stock |
|
| 100MG | 641 | In Stock |
|
| 200MG | 905 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product Name(E)-Akt inhibitor-IV
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NoteResearch use only, not for human use.
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Brief Description(E)-Akt inhibitor-IV ((E)-AKTIV) is an inhibitor of PI3K-Akt.
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Description(E)-Akt inhibitor-IV ((E)-AKTIV) is an inhibitor of PI3K-Akt.(In Vitro):(E)-Akt inhibitor-IV shows little effects on the growth of 184B5 non-cancer cells at the average GI20 doses.
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In Vitro——
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In Vivo——
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Synonyms(E)-Akt inhibitor-IV? | CS-1992 | (E)-AKTIV
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PathwayCytoskeleton/Cell Adhesion Molecules
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TargetAkt
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RecptormAChR
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Research Area——
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Indication——
Chemical Information
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CAS Number959841-49-7
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Formula Weight616.56
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Molecular FormulaC31H29IN4S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 50 mg/mL (81.36 mM)
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SMILESCCN(C1/C=C/N(C)c2ccccc2)c(cc(cc2)-c3nc(cccc4)c4s3)c2N1c1ccccc1.I
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Tran JA, et al. Differential coupling of muscarinic M1, M2, and M3 receptors to phosphoinositide hydrolysis in urinary bladder and longitudinal muscle of the ileum of the mouse. J Pharmacol Exp Ther. 2006 Aug;318(2):649-56. Epub 2006 May 4.
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