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Obafistat
CAS No. 2160582-57-8
Obafistat( —— )
Catalog No. M28228 CAS No. 2160582-57-8
Obafistat is a potent aldo-keto reductase AKR1C3 inhibitor with an IC 50 of 1.2 nM for human AKR1C3 .
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 28 | In Stock |
|
| 2MG | 45 | In Stock |
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| 5MG | 73 | In Stock |
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| 10MG | 113 | In Stock |
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| 25MG | 188 | In Stock |
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| 50MG | 300 | In Stock |
|
| 100MG | 485 | In Stock |
|
| 200MG | 668 | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameObafistat
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NoteResearch use only, not for human use.
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Brief DescriptionObafistat is a potent aldo-keto reductase AKR1C3 inhibitor with an IC 50 of 1.2 nM for human AKR1C3 .
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DescriptionObafistat is a potent aldo-keto reductase AKR1C3 inhibitor with an IC 50 of 1.2 nM for human AKR1C3 .
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayMembrane Transporter/Ion Channel
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TargetNADPH
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number2160582-57-8
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Formula Weight365.38
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Molecular FormulaC15H16FN5O3S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 62.5 mg/mL (171.05 mM)
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SMILESO=C(c1cnn[nH]1)N(CC1CC2)CC2N1S(c1cc(F)ccc1)(=O)=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Simonetta KR, et al. Prospective discovery of small molecule enhancers of an E3 ligase-substrate interaction. Nat Commun. 2019 Mar 29;10(1):1402.
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