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BML-259
CAS No. 267654-00-2
BML-259( CAY10554 )
Catalog No. M28107 CAS No. 267654-00-2
BML-259 is an inhibitor of CDK5 and CDK2 with IC50s of 64 and 98 nM, respectively. BML-259 can be used in studies about the treatment of cancer and neurodegenerative diseases.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 46 | In Stock |
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| 5MG | 41 | In Stock |
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| 10MG | 73 | In Stock |
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| 25MG | 163 | In Stock |
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| 50MG | 272 | In Stock |
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| 100MG | 477 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | 1014 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBML-259
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NoteResearch use only, not for human use.
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Brief DescriptionBML-259 is an inhibitor of CDK5 and CDK2 with IC50s of 64 and 98 nM, respectively. BML-259 can be used in studies about the treatment of cancer and neurodegenerative diseases.
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DescriptionBML-259 is an inhibitor of CDK5 and CDK2 with IC50s of 64 and 98 nM, respectively. BML-259 can be used in studies about the treatment of cancer and neurodegenerative diseases.(In Vitro):BML-259 prevents a large population of cells from NAC-evoked cell death.
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In VitroBML-259 (10 μM) protects large population of cells against non-Aβ component of Alzheimer's disease amyloid (NAC)-evoked cell death.
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In Vivo——
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SynonymsCAY10554
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PathwayAngiogenesis
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TargetCDK
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RecptorAntifungal|Antiviral
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Research Area——
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Indication——
Chemical Information
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CAS Number267654-00-2
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Formula Weight260.36
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Molecular FormulaC14H16N2OS
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (480.12 mM)
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SMILESO=C(NC1=NC=C(S1)C(C)C)CC=2C=CC=CC2
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Freitas-Silva O, et al. Tracing fungi secondary metabolites in Brazil nuts using LC-MS/MS. Drug Metab Lett. 2011 Aug;5(3):150-5.
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