Home - Products - Endocrinology/Hormones - Androgen Receptor (AR) - VPC-13566

VPC-13566

CAS No. 218464-59-6

VPC-13566( VPC13566 | VPC 13566 )

Catalog No. M27935 CAS No. 218464-59-6

VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket.

Purity : >98% (HPLC)

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

Size	Price / USD	Stock	Quantity
1 mL x 10 mM in DMSO	110	In Stock
5MG	93	In Stock
10MG	155	In Stock
25MG	276	In Stock
50MG	433	In Stock
100MG	651	In Stock
200MG	901	In Stock
500MG	Get Quote	In Stock
1G	Get Quote	In Stock

Get Quotation Bulk Inquiry Add to Cart

Biological Information

Product Name

VPC-13566
Note

Research use only, not for human use.
Brief Description

VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket.
Description

VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the BF3 pocket. VPC-13566 inhibits the growth of various prostate cancer cell lines and reduces the growth of AR-dependent prostate cancer xenograft tumors in mice.
In Vitro

——
In Vivo

——
Synonyms

VPC13566 | VPC 13566
Pathway

Endocrinology/Hormones
Target

Androgen Receptor (AR)
Recptor

——
Research Area

——
Indication

——

Chemical Information

CAS Number

218464-59-6
Formula Weight

258.324
Molecular Formula

C18H14N2
Purity

>98% (HPLC)
Solubility

In Vitro:?DMSO : 100 mg/mL (387.12 mM)
SMILES

Cc1cccc2c(c[nH]c12)-c1ccc2ccccc2n1
Chemical Name

——

Shipping & Storage Information

Storage

(-20℃)
Shipping

With Ice Pack
Stability

≥ 2 years

Reference

1.Anthony Boitano, et al. Aryl hydrocarbon receptor antagonists and methods of use thereof for treating various diseases. WO2020051207A2

Calculator

Molecular Weight Calculator

Dilution Calculator

Molarity Calculator

molnova catalog

related products

Oxandrolone

Oxandrolone(SC11585) is a synthetic hormone with anabolic and androgenic properties.
BMS-986365

BMS-986365 (CC-94676) is an orally available, selective and highly potent AR degrader with potential anticancer activity that inhibits AR signaling and suppresses tumor growth for the study of prostate cancer.
Testosterone Enantha...

Testosterone Enanthate is a long-acting intramuscular form of the androgen testosterone.

Sign In Join Free