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DDD85646
CAS No. 1215010-55-1
DDD85646( DDD-85646 | DDD 85646 )
Catalog No. M27869 CAS No. 1215010-55-1
DDD85646 is an inhibitor of T. brucei N-myristoyltransferase with a Ki of 1.44 nM, an IC50 of 2 nM and an EC50 of 2 nM. The IC50 of hNMT is 4 nM.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 291 | In Stock |
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| 5MG | 266 | In Stock |
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| 10MG | 400 | In Stock |
|
| 25MG | 676 | In Stock |
|
| 50MG | 921 | In Stock |
|
| 100MG | 1265 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameDDD85646
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NoteResearch use only, not for human use.
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Brief DescriptionDDD85646 is an inhibitor of T. brucei N-myristoyltransferase with a Ki of 1.44 nM, an IC50 of 2 nM and an EC50 of 2 nM. The IC50 of hNMT is 4 nM.
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DescriptionDDD85646 is an inhibitor of T. brucei N-myristoyltransferase with a Ki of 1.44 nM, an IC50 of 2 nM and an EC50 of 2 nM. The IC50 of hNMT is 4 nM.
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In Vitro——
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In Vivo——
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SynonymsDDD-85646 | DDD 85646
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PathwayMicrobiology/Virology
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TargetParasite
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RecptorGABAA
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Research Area——
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Indication——
Chemical Information
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CAS Number1215010-55-1
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Formula Weight495.42
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Molecular FormulaC21H24Cl2N6O2S
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 100 mg/mL (201.84 mM)
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SMILESCc1nn(C)c(C)c1NS(=O)(=O)c1c(Cl)cc(cc1Cl)-c1ccnc(c1)N1CCNCC1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Quan Z, et al. Reactive oxygen species-mediated endoplasmic reticulum stress and mitochondrial dysfunction contribute to cirsimaritin-induced apoptosis in human gallbladder carcinoma GBC-SD cells. Cancer Lett. 2010 Sep 28;295(2):252-9.
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