Ocinaplon

CAS No. 96604-21-6

Ocinaplon( DOV 273547 )

Catalog No. M27674 CAS No. 96604-21-6

Ocinaplon is a GABAA receptors modulator.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 28 In Stock
5MG 50 In Stock
10MG 88 In Stock
25MG 179 In Stock
50MG 261 In Stock
100MG 366 In Stock
200MG 535 In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Ocinaplon
  • Note
    Research use only, not for human use.
  • Brief Description
    Ocinaplon is a GABAA receptors modulator.
  • Description
    Ocinaplon is a GABAA receptors modulator.(In Vivo):In rats, ocinaplon produces significant muscle relaxation, ataxia, and sedation only at doses >25-fold higher than the minimum effective dose (3.1 mg/kg) in the Vogel "conflict" test.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    DOV 273547
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    P2X7
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    96604-21-6
  • Formula Weight
    301.309
  • Molecular Formula
    C17H11N5O
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 2 mg/mL (6.64 mM)
  • SMILES
    O=C(c1cnn2c(ccnc12)-c1ccncc1)c1ccccn1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Hopper AT, et al. Synthesis and Characterization of the Novel Rodent-Active and CNS-Penetrant P2X7 Receptor Antagonist Lu AF27139. J Med Chem. 2021;64(8):4891-4902.
molnova catalog
related products
  • Silybin B

    Silybin B is an effective inhibitor of raloxifene 4 '- and 6-glucosalylation, an effective anti-fibrinogenic and anti-oligomeric component of Silymarin, with free radical scavenging activity of 1, 1-diphenyl-2-pyridinyl hydrazine (DPPH), and a protective effect against cisplatin-induced neurotoxicity by alleviating DNA damage and apoptosis.

  • Dehydrovomifoliol

    Dehydrovomifoliol could be a marker of Polish heather honey. Dehydrovomifoliol exhibits moderate acetylcholinesterase (AChE) inhibitory activities.

  • 18α-Glycylrrhizin

    18α-Glycyrrhizic acid is a derivate of Glycyrrhizic acid. 18α-Glycyrrhizic acid has weak antihepatotoxic anti-inflammatory activities.