MEDICA16

CAS No. 87272-20-6

MEDICA16( MEDICA 16 )

Catalog No. M27653 CAS No. 87272-20-6

MEDICA16 is a selective agonist for GPR40 as well as a partial agonist for GPR120.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
1 mL x 10 mM in DMSO 73 In Stock
5MG 55 In Stock
10MG 84 In Stock
25MG 178 In Stock
50MG 299 In Stock
100MG 433 In Stock
200MG Get Quote In Stock
500MG 904 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    MEDICA16
  • Note
    Research use only, not for human use.
  • Brief Description
    MEDICA16 is a selective agonist for GPR40 as well as a partial agonist for GPR120.
  • Description
    MEDICA16 is a selective agonist for GPR40 as well as a partial agonist for GPR120. MEDICA16, an ATP-citrate lyase inhibitor, significantly reduces intracellular TG content in gastrocnemius muscle with an increase in insulin sensitivity.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    MEDICA 16
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    GPR
  • Recptor
    PHD3|HIF-2α|VEGFR1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    87272-20-6
  • Formula Weight
    342.52
  • Molecular Formula
    C20H38O4
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 100 mg/mL (291.96 mM)
  • SMILES
    CC(C)(CCCCCCCCCCC(C)(C)CC(O)=O)CC(O)=O
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Roda JM, et al. Stabilization of HIF-2α induces sVEGFR-1 production from tumor-associated macrophages and decreases tumor growth in a murine melanoma model. J Immunol. 2012 Sep 15;189(6):3168-77.
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