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CP94253 hydrochloride
CAS No. 845861-39-4
CP94253 hydrochloride( CP 94253 hydrochloride )
Catalog No. M27617 CAS No. 845861-39-4
CP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 1 mL x 10 mM in DMSO | 61 | In Stock |
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| 5MG | 61 | In Stock |
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| 10MG | 92 | In Stock |
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| 25MG | 217 | In Stock |
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| 50MG | 346 | In Stock |
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| 100MG | 555 | In Stock |
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| 200MG | 770 | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCP94253 hydrochloride
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NoteResearch use only, not for human use.
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Brief DescriptionCP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.
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DescriptionCP94253 hydrochloride is a potent, selective and centrally active agonist of 5-HT1B receptor with Ki of 2 nM. The Kis are 89, 49, 860, and 1600 nM for 5-HT1A, 5-HT1D, 5-HT1C and 5-HT2 receptors, respectively.
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In Vitro——
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In Vivo——
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SynonymsCP 94253 hydrochloride
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PathwayOthers
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TargetOther Targets
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Recptorpanx1|Topo IV|Bacterial|DNA-gyrase
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Research Area——
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Indication——
Chemical Information
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CAS Number845861-39-4
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Formula Weight293.8
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Molecular FormulaC15H20ClN3O
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 125 mg/mL (425.47 mM)
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SMILESCl.CCCOc1ccc2[nH]cc(C3=CCNCC3)c2n1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Poon IK, et al. Unexpected link between an antibiotic, pannexin channels and apoptosis. Nature. 2014 Mar 20;507(7492):329-34.
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