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Cinitapride
CAS No. 66564-14-5
Cinitapride( Cidine | Blaston | Cinmove | Cintapro | Paxapride | cinitapride tartrate )
Catalog No. M27395 CAS No. 66564-14-5
Cinitapride is a gastroprokinetic agent. It slows the actions of the muscles to reduce the symptoms of conditions such as acid reflux, delayed gastric emptying, and ulcer dyspepsia.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 149 | In Stock |
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| 10MG | 239 | In Stock |
|
| 25MG | 479 | In Stock |
|
| 50MG | 692 | In Stock |
|
| 100MG | 972 | In Stock |
|
| 200MG | Get Quote | In Stock |
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| 500MG | Get Quote | In Stock |
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| 1G | Get Quote | In Stock |
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Biological Information
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Product NameCinitapride
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NoteResearch use only, not for human use.
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Brief DescriptionCinitapride is a gastroprokinetic agent. It slows the actions of the muscles to reduce the symptoms of conditions such as acid reflux, delayed gastric emptying, and ulcer dyspepsia.
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DescriptionCinitapride is a gastroprokinetic agent. It slows the actions of the muscles to reduce the symptoms of conditions such as acid reflux, delayed gastric emptying, and ulcer dyspepsia. Cinitapride acts as an antagonist of the 5-HT2 receptors and as an agonist of the 5-HT1 and 5-HT4 receptors.
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In Vitro——
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In VivoCinitapride (intraperitoneal injection; 0.25-1 mg/kg; once) shows gastroprotective effetcs in gastric ulceration rat model. Animal Model:Male Wistar rats with gastric ulcerationDosage:0.25-1 mg/kg Administration:Intraperitoneal injection; 0.25-1 mg/kg; once Result:Reduced haemorrhagic lesions compared with the ulcerated control group.Decreased the percentage of ulceration to 28.76% at the highest dose (1 mg/kg).Attenuated the increase myeloperoxidase activity (p<0.05, p<0.01).Increased GSH-px activity in the gastric mucosa.
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SynonymsCidine | Blaston | Cinmove | Cintapro | Paxapride | cinitapride tartrate
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PathwayEndocrinology/Hormones
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Target5-HT Receptor
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Recptor——
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Research Area——
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Indication——
Chemical Information
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CAS Number66564-14-5
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Formula Weight402.495
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Molecular FormulaC21H30N4O4
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Purity>98% (HPLC)
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SolubilityIn Vitro:?DMSO : 20.83 mg/mL (51.75 mM)
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SMILESCCOc1cc(N)c(cc1C(=O)NC1CCN(CC2CCC=CC2)CC1)[N+]([O-])=O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Feng N, et, al. Amides produced by Streptoverticillium morookaense. SAGE Journals. 2007 Jan; 2(2):151-153.
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