ZEN-3862

CAS No. 1952264-33-3

ZEN-3862( ZEN 3862 | ZEN3862 )

Catalog No. M26520 CAS No. 1952264-33-3

ZEN-3862 is an inhibitor of BET(IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 125 Get Quote
5MG 205 Get Quote
10MG 320 Get Quote
25MG 565 Get Quote
50MG 799 Get Quote
100MG 1071 Get Quote
500MG 2151 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    ZEN-3862
  • Note
    Research use only, not for human use.
  • Brief Description
    ZEN-3862 is an inhibitor of BET(IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively).
  • Description
    ZEN-3862 is an inhibitor of BET(IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively). ZEN-3862 can be used to form PROTACs to induce degradation of BRD4.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ZEN 3862 | ZEN3862
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    ——
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1952264-33-3
  • Formula Weight
    340.354
  • Molecular Formula
    C19H17FN2O3
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : 83.33 mg/mL (244.84 mM)
  • SMILES
    Cc1noc(C)c1-c1ccc(=O)n(Cc2ccc(C3CO3)c(F)c2)c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Sikorska H, et al. [Physiological functions of L-ornithine and L-aspartate in the body and the efficacy of administration of L-ornithine-L-aspartate in conditions of relative deficiency]. Pol Merkur Lekarski. 2010 Jun;28(168):490-5.
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