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PF-06821497
CAS No. 1844849-10-0
PF-06821497( —— )
Catalog No. M26370 CAS No. 1844849-10-0
PF-06821497 is a selective inhibitor of EZH2 with significant tumor growth inhibition.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 393 | Get Quote |
|
| 10MG | 581 | Get Quote |
|
| 25MG | 888 | Get Quote |
|
| 50MG | 1242 | Get Quote |
|
| 100MG | 1674 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NamePF-06821497
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NoteResearch use only, not for human use.
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Brief DescriptionPF-06821497 is a selective inhibitor of EZH2 with significant tumor growth inhibition.
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DescriptionPF-06821497 is a selective inhibitor of EZH2 with significant tumor growth inhibition.(In Vivo):The tumor regression effect of PF-06821497 can be sustained for another 40 days.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayChromatin/Epigenetic
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TargetHistone Demethylase
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RecptorApoptosis| Autophagy
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Research Area——
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Indication——
Chemical Information
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CAS Number1844849-10-0
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Formula Weight467.34
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Molecular FormulaC22H24Cl2N2O5
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Purity>98% (HPLC)
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Solubility——
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SMILESCO[C@H](C1COC1)c1cc(Cl)c2CCN(Cc3c(OC)cc(C)[nH]c3=O)C(=O)c2c1Cl
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Greim H, Saltmiras D, Mostert V, Strupp C. Evaluation of carcinogenic potential of the herbicide glyphosate, drawing on tumor incidence data from fourteen chronic/carcinogenicity rodent studies. Crit Rev Toxicol. 2015 Mar;45(3):185-208.
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